<p>Advanced Blood-Brain Barrier Drug Delivery is a reprint with a summary editorial followed by 16 chapters that cover five areas of brain drug delivery including receptor-mediated transport (RMT) carrier-mediated transport (CMT) active efflux transport (AET) Trojan horse lipid nanoparticles (LNP) and in vivo methods for measurement of drug transport across the blood-brain barrier (BBB).</p>